SCHEMBL7433457

SCHEMBL7433457

O=C(O)CCCCc1nc2ccccc2[nH]1

nearest known ligand 0.80

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 1/20 0.80
POLB P06746 1/20 0.73
CYP1A2 P05177 1/20 0.62
CYP2C9 P11712 1/20 0.62
KDM4E B2RXH2 1/20 0.59
MAPT P10636 2/20 0.59
ALDH1A1 P00352 1/20 0.59
NPC1 O15118 1/20 0.58
RAB9A P51151 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565997 0.98 CHRM1 (0.78) CHRM1POLBCYP1A2CYP2C9KDM4E
SCHEMBL2017763 0.95 CHRM1 (0.82) CHRM1POLBCYP1A2CYP2C9KDM4E
Procodazole SCHEMBL349966 0.89 CHRM1 (1.00) CHRM1POLBCYP1A2CYP2C9KDM4E
Procodazole SCHEMBL29404024 0.89 CHRM1 (1.00) CHRM1POLBCYP1A2CYP2C9KDM4E
Procodazole SCHEMBL838841 0.89 CHRM1 (1.00) CHRM1POLBCYP1A2CYP2C9KDM4E
SCHEMBL1231977 0.85 GAA (0.76) CHRM1KDM4EMAPTALDH1A1
SCHEMBL7006523 0.85 POLB (1.00) CHRM1POLBNPC1RAB9A
Procodazole SCHEMBL5413283 0.85 CHRM1 (0.91) CHRM1POLBCYP1A2CYP2C9KDM4E
SCHEMBL721483 0.84 HDAC3 (0.70) CHRM1POLBKDM4E
SCHEMBL718972 0.84 HDAC3 (0.70) CHRM1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5140011-A Hypotensive agents HOFFMANN-LA ROCHE, INC. (US) 1992-08-18 US disclosed
EP-0391179-A2 Peptide derivatives of amino acids having a renin-inhibiting effect F. HOFFMANN-LA ROCHE AG (CH) 1990-10-10 EP disclosed