SCHEMBL7433472

SCHEMBL7433472

O=C(O)CCc1cc(C2CCCN2C(=O)Cc2ccc(OCc3ccc(F)cc3)cc2)no1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CPT1A P50416 1/20 0.42
FFAR1 O14842 7/20 0.42
HRH3 Q9Y5N1 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GRM5 P41594 2/20 0.41
AADAT Q8N5Z0 1/20 0.39
FFAR4 Q5NUL3 2/20 0.39
BTK Q06187 2/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
YAP1 P46937 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481567 0.93 FFAR1 (0.45) FFAR1HRH3AADATFFAR4YAP1
SCHEMBL7433078 0.92 FFAR1 (0.42) CPT1AFFAR1HRH3AADATFFAR4
SCHEMBL7435979 0.92 CPT1A (0.43) CPT1AFFAR1HRH3SMN1; SMN2FFAR4
SCHEMBL7542862 0.92 CPT1A (0.42) CPT1AFFAR1FFAR4RXRARXRB
SCHEMBL7487553 0.92 FFAR1 (0.42) CPT1AFFAR1HRH3AADATFFAR4
SCHEMBL7583778 0.87 FFAR1 (0.44) FFAR1SMN1; SMN2FFAR4
SCHEMBL7488778 0.87 FFAR1 (0.47) FFAR1GRM5AADATFFAR4YAP1
SCHEMBL7427523 0.86 NPC1 (0.49) CPT1AFFAR1FFAR4
SCHEMBL7484778 0.86 FFAR1 (0.45) CPT1AFFAR1AADATFFAR4
SCHEMBL7434473 0.86 NPC1 (0.45) CPT1AFFAR1BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244656-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES Pfizer Products Inc. (US) 2002-10-02 EP disclosed
WO-2001051487-A1 NON-PEPTIDYL INHIBITORS OF VLA-4 DEPENDENT CELL BINDING USEFUL IN TREATING INFLAMMATORY, AUTOIMMUNE, AND RESPIRATORY DISEASES PFIZER PRODUCTS INC. (US) 2001-07-19 WO disclosed