SCHEMBL7433753

SCHEMBL7433753

COc1cc(CC(=O)N2CCC(CNC(=O)N3CCC(C(=O)O)CC3)CC2)ccc1NC(=O)Nc1ccccc1C

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 14/20 0.54
ITGB1 P05556 10/20 0.54
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
KMT2A Q03164 1/20 0.46
ATM Q13315 1/20 0.46
POLB P06746 1/20 0.44
L3MBTL1 Q9Y468 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7432187 0.95 ITGA4 (0.52) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7429260 0.92 ITGA4 (0.54) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7430255 0.86 ITGA4 (0.60) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7427700 0.85 ITGA4 (0.54) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7423889 0.85 ITGA4 (0.54) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7434801 0.85 ITGA4 (0.55) ITGA4ITGB1
SCHEMBL7425325 0.84 ITGA4 (0.54) ITGA4ITGB1
SCHEMBL7424393 0.83 ITGA4 (0.53) ITGA4ITGB1MEN1ALDH1A1KMT2A
SCHEMBL7388473 0.82 ITGA4 (0.59) ITGA4ITGB1
SCHEMBL7389620 0.82 ITGA4 (0.53) ITGA4ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1999054321-A1 SUBSTITUTED DIAMINES AND THEIR USE AS CELL ADHESION INHIBITORS AVENTIS PHARMA LIMITED (GB) 1999-10-28 WO disclosed