SCHEMBL7433869

SCHEMBL7433869

COC(=O)CCCCCc1ccc(C#N)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CYP11B1 P15538 1/20 0.52
CYP11B2 P19099 1/20 0.52
HPGD P15428 1/20 0.46
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 1/20 0.44
FAAH O00519 1/20 0.44
EPHX2 P34913 1/20 0.43
HTT P42858 2/20 0.43
PDE3B Q13370 1/20 0.43
PDE3A Q14432 1/20 0.43
P2RY12 Q9H244 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.42
SAE1 Q9UBE0 1/20 0.42
UBA2 Q9UBT2 1/20 0.42
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1337450 0.94 CYP11B1 (0.54) TSHRHSD17B10CYP11B1CYP11B2POLB
SCHEMBL1338556 0.87 CYP11B1 (0.60) CYP11B1CYP11B2POLBMAPTHTT
SCHEMBL22146949 0.85 HPGD (0.46) TSHRHPGDEPHX2PDE3BPDE3A
SCHEMBL27537788 0.83 TSHR (0.46) TSHRHSD17B10CYP11B1CYP11B2HDAC1
SCHEMBL3628694 0.83 CYP11B1 (0.56) TSHRHSD17B10CYP11B1CYP11B2HPGD
SCHEMBL21169244 0.83 TSHR (0.57) TSHRHSD17B10MAPTHDAC1FAAH
SCHEMBL20717646 0.82 FFAR1 (0.61) MAPTHDAC1HDAC2
Hydrochloric Acid SCHEMBL3628690 0.82 CYP11B1 (0.55) TSHRHSD17B10CYP11B1CYP11B2HPGD
SCHEMBL29165966 0.81 FFAR1 (0.48) HDAC1FAAHPDE3BPDE3AP2RY12
SCHEMBL25169991 0.81 FAAH (0.59) HSD17B10MAPTFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0725059-B1 2,3-DIAMINOPROPIONIC ACID DERIVATIVE SUMITOMO PHARMA (JP) 2001-01-17 EP disclosed
US-6048854-A ANTICOAGULANTS; ANTICANCER AGENT; WOUND HEALING AGENTS;BONE DISORDERS SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 2000-04-11 US disclosed
US-5707994-A USEFUL AS A PLATELET AGGREGATION INHIBITOR, CANCER METASTASIS INHIBITOR, WOUND HEALING AGENT OR A BONE RESORPTION INHIBITOR SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-01-13 US disclosed
EP-0502536-B1 Phenyl amidines derivatives useful as platelet aggregation inhibitors SEARLE & CO (US) 1996-10-09 EP disclosed
EP-0725059-A1 2,3-DIAMINOPROPIONIC ACID DERIVATIVE SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1996-08-07 EP disclosed
US-5481021-A Phenyl amidines derivatives useful as platelet aggregation inhibitors G. D. SEARLE & CO. (US) 1996-01-02 US disclosed
EP-0574545-B1 PHENYL AMIDINES DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS SEARLE & CO (US) 1994-11-30 EP disclosed
EP-0574545-A1 PHENYL AMIDINES DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS. SEARLE & CO (US) 1993-12-22 EP disclosed
WO-1992015607-A2 PHENYL AMIDINES DERIVATIVES USEFUL AS PLATELET AGGREGATION INHIBITORS G.D. SEARLE & CO. (US) 1992-09-17 WO disclosed
EP-0502536-A1 Phenyl amidines derivatives useful as platelet aggregation inhibitors G.D. Searle & Co. (US) 1992-09-09 EP disclosed