SCHEMBL7434320

SCHEMBL7434320

CC(C)C[CH]C(=O)N([C@H]1CCCNCC1=O)S(=O)(=O)c1cccc(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 2/20 0.36
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HSD11B1 P28845 2/20 0.34
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
HSD11B2 P80365 1/20 0.34
GHSR Q92847 8/20 0.34
HTT P42858 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424733 0.89 PSEN1 (0.44) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7426764 0.88 KCNA5 (0.39) KCNA5HSD11B1PSEN1PSEN2APH1B
SCHEMBL7434860 0.88 KCNA5 (0.39) KCNA5HSD11B1PSEN1PSEN2APH1B
SCHEMBL7434329 0.81 KCNA5 (0.35) KCNA5SLC6A2SLC6A4SLC6A3HTR2A
SCHEMBL4765458 0.81 HTR6 (0.40) KCNA5SLC6A2SLC6A3HTR2AHTR2C
SCHEMBL4762983 0.81 PSEN1 (0.36) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL6590944 0.80 PSEN1 (0.31) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL4761958 0.80 PSEN1 (0.31) PSEN1PSEN2APH1BNCSTNAPH1A
SCHEMBL7433037 0.79
SCHEMBL4761916 0.79 PSEN1 (0.33) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed