SCHEMBL7435213

SCHEMBL7435213

COC(=O)CNc1ccccc1C(=O)OC

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.66
GLA P06280 1/20 0.66
KMT2A Q03164 2/20 0.62
MEN1 O00255 1/20 0.62
NPC1 O15118 1/20 0.62
POLB P06746 2/20 0.61
ATM Q13315 1/20 0.61
ALDH1A1 P00352 7/20 0.58
HTT P42858 1/20 0.58
MAPT P10636 3/20 0.56
ALOX15 P16050 1/20 0.56
GAA P10253 4/20 0.54
LMNA P02545 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
HSD17B10 Q99714 5/20 0.51
ADRA1D P25100 1/20 0.51
ADRA1A P35348 1/20 0.51
ADRA1B P35368 1/20 0.51
TSHR P16473 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7528637 0.87 KDM4E (0.71) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL5807758 0.86 KDM4E (0.49) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL2707530 0.86 KDM4E (0.66) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL7878306 0.86 KDM4E (0.57) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL7873424 0.86 ADRA1A (0.54) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL7434506 0.86 KDM4E (0.57) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL8047226 0.85 KMT2A (0.56) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL6318031 0.84 KDM4E (0.72) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL7875568 0.84 KDM4E (0.55) KDM4EGLAKMT2AMEN1NPC1
SCHEMBL7875557 0.84 KDM4E (0.55) KDM4EGLAKMT2AMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113768936-B Application of evodiamine derivative in preparation of medicine for treating superficial fungal infection 南华大学 2023-04-14 CN disclosed
CN-113768936-A Application of evodiamine derivative in preparation of medicine for treating superficial fungal infection 南华大学 2021-12-10 CN disclosed
US-20020091148-A1 3-substituted indole antiproliferative angiogenesis inhibitors ABBOTT LABORATORIES 2002-07-11 US disclosed
WO-2002022576-A2 3-SUBSTITUTED INDOLE CARBOHYDRAZIDES USEFUL AS CELL PROLIFERATION AND ANGIOGENESIS INHIBITORS ABBOTT LABORATORIES (US) 2002-03-21 WO disclosed
US-6001831-A Process for producing quinazoline derivatives CLARIANT GMBH (DE) 1999-12-14 US disclosed
EP-0847392-B1 PROCESS FOR PRODUCING QUINAZOLINE DERIVATIVES CLARIANT GMBH (DE) 1999-12-08 EP disclosed
EP-0738258-B1 PROCESS FOR PREPARING N-SUBSTITUTED GLYCINIC ACIDS OR GLYCINE ESTERS AND USE OF SAID PROCESS IN INDIGO SYNTHESIS DSM FINE CHEM AUSTRIA GMBH (AT) 1999-07-28 EP disclosed
CN-1194639-A Quinazoline derivatives and their use as anti-inflammatory agents CORIEN CO LTD (DE) 1998-09-30 CN disclosed
EP-0640594-A1 Hydantoin derivative as metalloprotease inhibitor FUJIREBIO INC. (JP) 1995-03-01 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020091148-A1 3-substituted indole antiproliferative angiogenesis inhibitors MKI67, FLT4, IDO1 KDM4E 1608/4885GLA 1576/4885KMT2A 2765/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.