SCHEMBL7435263

SCHEMBL7435263

COc1cccc(C(=O)NC2CC3CCC(C2)N3C)c1C

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 5/20 0.63
HSP90AB1 P08238 5/20 0.63
HTR4 Q13639 1/20 0.57
HTR3A P46098 3/20 0.56
CYP3A4 P08684 1/20 0.56
KCNH2 Q12809 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3165934 0.84 TAS1R3 (0.67) HSP90AA1HSP90AB1
SCHEMBL14817133 0.80 TAS1R3 (0.76) HSP90AA1HSP90AB1
SCHEMBL9732092 0.80
SCHEMBL2427286 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2425089 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2425092 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2426001 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2426003 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2427289 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1
SCHEMBL2423578 0.79 HSP90AA1 (0.85) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5491148-A TREATING GASTROINTESTINAL, CARDIOVASCULAR, CENTRAL NERVOUS SYSTEM DISORDERS, EMESIS, PAIN SYNTEX (U.S.A.) INC. (US) 1996-02-13 US disclosed