SCHEMBL7435996

SCHEMBL7435996

CC(C)[C@H](NC(=O)N(C)Cc1cscn1)C(=O)NC(Cc1ccccc1)C(O)[C@H](O)[C@H](Cc1ccccc1)NC(=O)[C@@H](NC(=O)N(C)Cc1cscn1)C(C)C

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.74
CYP3A4 P08684 17/20 0.60
CYP2D6 P10635 5/20 0.52
CYP2C19 P33261 3/20 0.52
CYP1A2 P05177 2/20 0.52
CYP2C9 P11712 3/20 0.47
MEN1 O00255 1/20 0.47
SLC22A2 O15244 1/20 0.47
SLC22A1 O15245 1/20 0.47
ABCC3 O15438 1/20 0.47
ABCC4 O15439 1/20 0.47
MLNR O43193 1/20 0.47
NR1I2 O75469 1/20 0.47
SLCO2B1 O94956 1/20 0.47
ABCB11 O95342 1/20 0.47
ALDH1A1 P00352 1/20 0.47
PGR P06401 1/20 0.47
ABCB1 P08183 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436001 1.00 CA2 (0.74) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7340732 1.00 CA2 (0.74) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7343373 1.00 CA2 (0.74) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7339666 1.00 CA2 (0.74) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7339424 0.95 CA2 (0.67) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7334177 0.95 CA2 (0.84) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7338296 0.92 CA2 (0.63) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7336293 0.89 CA2 (0.61) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7298756 0.89 CA2 (0.77) CA2CYP3A4CYP2D6CYP2C19CYP1A2
SCHEMBL7342547 0.86 CA2 (0.57) CA2CYP3A4CYP2D6CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0486948-A2 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1992-05-27 EP disclosed