SCHEMBL7436134

SCHEMBL7436134

CCCCC(NCC(CC(C)C)NC(=O)c1ccc(F)c(C(F)(F)F)c1)C(=O)CSCc1ccco1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 3/20 0.36
ALDH1A1 P00352 3/20 0.36
USP2 O75604 1/20 0.36
MAPT P10636 1/20 0.36
HSD17B10 Q99714 1/20 0.36
TAS1R3 Q7RTX0 6/20 0.33
TAS1R1 Q7RTX1 6/20 0.33
HDAC8 Q9BY41 1/20 0.32
TAS1R2 Q8TE23 1/20 0.32
TRPV1 Q8NER1 2/20 0.32
HPGD P15428 1/20 0.32
TP53 P04637 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
TSHR P16473 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7310667 0.92 ALDH1A1 (0.39) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL8686162 0.90 NPC1 (0.48) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7436141 0.88 NPC1 (0.38) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7304180 0.88 NPC1 (0.38) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7300617 0.88 ALDH1A1 (0.37) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7313603 0.88 ALDH1A1 (0.40) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7429973 0.88 ALDH1A1 (0.35) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL8681390 0.87 CYP1A2 (0.36) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7310588 0.87 HPGD (0.41) NPC1RAB9APOLBALDH1A1USP2
SCHEMBL7306338 0.87 ALDH1A1 (0.38) NPC1RAB9APOLBALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed