SCHEMBL743627

SCHEMBL743627

COc1ccc(C=CC(=O)c2c(OC)cc(OC)c(CN3CCCCC3)c2O)cc1

nearest known ligand 0.83

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 8/20 0.65
TDP1 Q9NUW8 1/20 0.57
ABCG2 Q9UNQ0 2/20 0.55
SLC5A1 P13866 1/20 0.52
SLC5A2 P31639 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3706909 1.00 ABCB1 (0.65) ABCB1TDP1ABCG2SLC5A1SLC5A2
SCHEMBL20858974 0.92 ABCB1 (0.57) ABCB1TDP1ABCG2SLC5A1SLC5A2
SCHEMBL746760 0.92 ABCB1 (0.54) ABCB1
SCHEMBL745647 0.92 ABCB1 (0.54) ABCB1
SCHEMBL7030048 0.91 ABCB1 (0.53) ABCB1
SCHEMBL13075312 0.90 ABCB1 (0.56) ABCB1TDP1ABCG2SLC5A1SLC5A2
SCHEMBL7028459 0.90 ABCB1 (0.56) ABCB1TDP1ABCG2SLC5A1SLC5A2
SCHEMBL742054 0.90 ABCB1 (0.63) ABCB1TDP1ABCG2
SCHEMBL746215 0.89 ABCB1 (0.67) ABCB1ABCG2
SCHEMBL7030123 0.85 ABCB1 (0.57) ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429292-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER Georgia State University Research Foundation, Inc. (US) 2012-03-21 EP claimed
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO claimed
EP-2429292-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER Georgia State University Research Foundation, Inc. (US) 2012-03-21 EP disclosed
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO disclosed