SCHEMBL745647

SCHEMBL745647

COc1cc(OC)c(C(=O)C=Cc2ccc(C)cc2)c(O)c1CN1CCCCC1

nearest known ligand 0.83

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 10/20 0.54
MAPT P10636 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
PDPK1 O15530 1/20 0.49
TTR P02766 1/20 0.49
ALOX5 P09917 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL746760 1.00 ABCB1 (0.54) ABCB1MAPTNPSR1PDPK1TTR
SCHEMBL20858964 0.93 ABCB1 (0.49) ABCB1MAPTNPSR1PDPK1TTR
SCHEMBL3706909 0.92 ABCB1 (0.65) ABCB1
SCHEMBL743627 0.92 ABCB1 (0.65) ABCB1
SCHEMBL7030048 0.91 ABCB1 (0.53) ABCB1MAPTNPSR1
SCHEMBL7028453 0.90 ABCB1 (0.47) ABCB1MAPTNPSR1PDPK1TTR
SCHEMBL744489 0.90 ABCB1 (0.56) ABCB1MAPT
SCHEMBL7030123 0.89 ABCB1 (0.57) ABCB1
SCHEMBL20858974 0.86 ABCB1 (0.57) ABCB1MAPTPDPK1TTRALOX5
SCHEMBL20858975 0.85 ABCB1 (0.47) ABCB1MAPTNPSR1PDPK1TTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429292-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER Georgia State University Research Foundation, Inc. (US) 2012-03-21 EP claimed
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO claimed
EP-2429292-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER Georgia State University Research Foundation, Inc. (US) 2012-03-21 EP disclosed
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO disclosed