SCHEMBL7437843

SCHEMBL7437843

COc1cc(CO)ccc1OCCCN1CCC(C(C#N)(c2ccc(F)cc2)c2ccc(F)cc2)C1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HRH3 Q9Y5N1 4/20 0.42
HTR1A P08908 4/20 0.42
DRD2 P14416 4/20 0.42
HTR2A P28223 4/20 0.42
MAPK1 P28482 1/20 0.41
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ABCB11 O95342 1/20 0.38
CHRM2 P08172 1/20 0.38
ADRA2A P08913 1/20 0.38
CHRM1 P11229 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
DRD1 P21728 1/20 0.38
DRD4 P21917 1/20 0.38
ACHE P22303 1/20 0.38
SLC6A2 P23975 1/20 0.38
HTR2C P28335 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7440743 0.95 KDM4E (0.46) KDM4EALDH1A1HRH3HTR1ADRD2
SCHEMBL7441509 0.88 KDM4E (0.45) KDM4EALDH1A1HRH3HTR1ADRD2
SCHEMBL7435551 0.87 KDM4E (0.43) KDM4EALDH1A1HRH3HTR1ADRD2
SCHEMBL7437790 0.87 ABCB11 (0.45) KDM4EALDH1A1HTR1ADRD2HTR2A
SCHEMBL10459160 0.86 ABCB11 (0.53) KDM4EALDH1A1HTR1ADRD2HTR2A
SCHEMBL7432347 0.86 KCNH2 (0.45) KDM4EALDH1A1HTR1ADRD2HTR2A
SCHEMBL7436121 0.85 HRH1 (0.45) HTR1ADRD2HTR2AABCB11CHRM2
SCHEMBL7435875 0.85 ABCB11 (0.45) KDM4EALDH1A1HTR1ADRD2HTR2A
SCHEMBL7432278 0.82 ABCB11 (0.44) ALDH1A1HTR1ADRD2HTR2AABCB11
SCHEMBL7438495 0.82 KDM4E (0.43) KDM4EALDH1A1HRH3HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5070087-A Aryl(alkyland alkylene)-N-((phenoxy and phenylthio)alkyl) aminoheterocyclics as cardiovascular, anthihistaminic, antisecretory and antiallergy agents A. H. ROBINS COMPANY, INCORPORATED (US) 1991-12-03 US disclosed