SCHEMBL743833

SCHEMBL743833

COc1cc(C(=O)O)c(CBr)c(Br)c1OC

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.51
FYN P06241 1/20 0.51
PTPN1 P18031 1/20 0.51
CA1 P00915 8/20 0.51
CA2 P00918 8/20 0.51
PKM P14618 1/20 0.47
HSD17B10 Q99714 2/20 0.45
CA9 Q16790 2/20 0.44
CA12 O43570 1/20 0.44
CA4 P22748 2/20 0.42
CA6 P23280 2/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
TPMT P51580 1/20 0.41
MAPT P10636 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
TSHR P16473 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL438401 0.86 KDM4E (0.53) PTPN1CA1CA2HSD17B10CA9
SCHEMBL14954265 0.82 PTPN1 (0.68) LCKFYNPTPN1CA1CA2
SCHEMBL30740970 0.79 LCK (0.56) LCKFYNPTPN1CA1CA2
SCHEMBL437132 0.79 LCK (0.56) LCKFYNPTPN1CA1CA2
SCHEMBL4302772 0.78 LCK (0.59) LCKFYNPTPN1PKMHSD17B10
SCHEMBL11541569 0.78 PKM (0.50) LCKFYNPTPN1PKMHSD17B10
SCHEMBL4551834 0.76 PKM (0.54) LCKFYNPKMHSD17B10ALDH1A1
SCHEMBL12497067 0.76 LCK (0.56) LCKFYNPTPN1PKMHSD17B10
SCHEMBL18280365 0.74 MAPT (0.56) LCKFYNCA1CA2HSD17B10
SCHEMBL7348961 0.74 MAPT (0.60) LCKFYNCA1CA2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429987-A2 AMIDE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING SAME Korea Research Institute Of Chemical Technology (KR) 2012-03-21 EP disclosed
WO-2010131922-A2 AMIDE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2010-11-18 WO disclosed