SCHEMBL7438374

SCHEMBL7438374

CC(C)C[C@H](NC(=O)OC[C@@H]1CCCO1)C(=O)NC(Cc1ccccc1)C(=O)CSCc1ccco1

nearest known ligand 0.54

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CAPN1 P07384 7/20 0.44
CYP1A2 P05177 1/20 0.42
CTSK P43235 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7438369 1.00 CAPN1 (0.44) CAPN1CYP1A2CTSK
SCHEMBL7438387 1.00 CAPN1 (0.44) CAPN1CYP1A2CTSK
SCHEMBL7438392 1.00 CAPN1 (0.44) CAPN1CYP1A2CTSK
SCHEMBL7305812 0.98 CAPN1 (0.43) CAPN1CTSK
SCHEMBL7305799 0.98 CAPN1 (0.43) CAPN1CTSK
SCHEMBL7305818 0.98 CAPN1 (0.43) CAPN1CTSK
SCHEMBL8683255 0.98 CAPN1 (0.43) CAPN1CTSK
SCHEMBL7437245 0.89 CAPN1 (0.46) CAPN1CTSK
SCHEMBL7437237 0.89 CAPN1 (0.46) CAPN1CTSK
SCHEMBL7438379 0.88 CYP1A2 (0.39) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed