SCHEMBL7439845

SCHEMBL7439845

CCc1cc(Cl)n2nc(-c3ccccc3)cc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.51
RAB9A P51151 7/20 0.51
ALDH1A1 P00352 4/20 0.51
SMN1; SMN2 Q16637 4/20 0.51
HPGD P15428 3/20 0.51
HTT P42858 2/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
KDM4E B2RXH2 6/20 0.50
MAPT P10636 3/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
GAA P10253 2/20 0.48
LMNA P02545 2/20 0.45
TP53 P04637 1/20 0.44
HSD17B10 Q99714 1/20 0.44
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
DPP4 P27487 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7436883 0.82 MAPT (0.52) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL7063800 0.80 RAB9A (0.71) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL13263646 0.80 NPC1 (0.53) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL7066066 0.77 HPGD (0.54) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL3559993 0.74 HSD17B10 (0.58) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL13501409 0.73 NPC1 (0.47) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL7842532 0.73 NPC1 (0.62) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL3299677 0.73 TP53 (0.53) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL311906 0.72 TP53 (0.47) NPC1RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL31417102 0.72 GRIN1 (0.38) TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed
EP-0579496-A1 4-Aminoquinazoline derivatives, and their use as medicine ONO PHARMACEUTICAL CO., LTD. (JP) 1994-01-19 EP disclosed