SCHEMBL7440755

SCHEMBL7440755

COC(=O)c1ccc(-c2c3nn(-c4ccc(Cl)cc4)c(=O)c-3c[nH]c2C)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.42
MAPT P10636 2/20 0.42
PSD A5PKW4 1/20 0.41
TP53 P04637 1/20 0.40
MAP2K4 P45985 1/20 0.40
DHODH Q02127 1/20 0.39
OPRM1 P35372 1/20 0.39
NPBWR1 P48145 1/20 0.39
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
KDM4A O75164 1/20 0.39
PTGS1 P23219 1/20 0.38
PTGS2 P35354 1/20 0.38
ALDH1A1 P00352 3/20 0.38
HPGD P15428 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
DRD2 P14416 1/20 0.38
TBXA2R P21731 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2649769 0.89 DHODH (0.44) MAPTDHODHNPSR1
SCHEMBL2649657 0.88 GAA (0.44) POLBMAPTPTGS1PTGS2ALDH1A1
Hydrochloric Acid SCHEMBL2662079 0.87 GAA (0.43) POLBMAPTPTGS1PTGS2ALDH1A1
SCHEMBL2648330 0.85 PTGS2 (0.45) MAPTNPBWR1PTGS1PTGS2HPGD
SCHEMBL2649535 0.85 GAA (0.43) MAPTTP53PTGS1PTGS2ALDH1A1
Hydrochloric Acid SCHEMBL2662511 0.85 PTGS2 (0.44) MAPTNPBWR1PTGS1PTGS2HPGD
SCHEMBL2650198 0.84 PSD (0.42) POLBMAPTPSDPTGS2ALDH1A1
SCHEMBL2650368 0.83 GAA (0.40) POLBMAPTPTGS1PTGS2ALDH1A1
SCHEMBL2649011 0.83 GAA (0.40) POLBMAPTPSDPTGS2ALDH1A1
SCHEMBL2648540 0.83 GAA (0.40) POLBMAPTPSDPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6333336-B1 GAMMA-AMINOBUTYRIC ACID RECEPTORS AS ANTICONVULSANTS FORMING THE COMPOUND BY AMIDATION MERCK SHARP & DOHME LTD. (GB) 2001-12-25 US disclosed