SCHEMBL7442980

SCHEMBL7442980

c1ccc2c(Cc3ccc(OCCN4CCCC4)cc3)c(-c3ccc(OCCN4CCCC4)cc3)oc2c1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 12/20 0.58
PSMB1 P20618 1/20 0.55
PSMB5 P28074 1/20 0.55
PSMB2 P49721 1/20 0.55
PTPN1 P18031 2/20 0.52
ESR1 P03372 4/20 0.51
ESR2 Q92731 3/20 0.51
HRH3 Q9Y5N1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6744827 0.94 LTA4H (0.60) LTA4HPSMB1PSMB5PSMB2PTPN1
Hydrochloric Acid SCHEMBL6749948 0.93 LTA4H (0.58) LTA4HPSMB1PSMB5PSMB2PTPN1
Hydrochloric Acid SCHEMBL6746982 0.93 ESR1 (0.59) LTA4HPSMB1PSMB5PSMB2ESR1
SCHEMBL6748810 0.84 ESR1 (0.63) PTPN1ESR1ESR2
SCHEMBL6748780 0.84 LTA4H (0.56) LTA4HPSMB1PSMB5PSMB2ESR1
SCHEMBL6744378 0.84 ESR1 (0.58) LTA4HPTPN1ESR1ESR2
SCHEMBL6745462 0.83 ESR1 (0.61) LTA4HPSMB1PSMB5PSMB2ESR1
Hydrochloric Acid SCHEMBL6749894 0.83 ESR1 (0.59) LTA4HPTPN1ESR1ESR2
Hydrochloric Acid SCHEMBL6745263 0.83 LTA4H (0.55) LTA4HPSMB1PSMB5PSMB2ESR1
Hydrochloric Acid SCHEMBL6751611 0.83 ESR1 (0.66) PTPN1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265575-B1 THROMBIN INHIBITORS ELI LILLY AND COMPANY 2001-07-24 US disclosed
US-6251921-B1 ADMINISTERING THROMBIN INHIBITING DIAMINE COMPOUND TO MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
US-6025382-A Antithrombotic diamines ELI LILLY AND COMPANY (US) 2000-02-15 US disclosed
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed