SCHEMBL7443540

SCHEMBL7443540

COC(=O)c1ccc(C)nc1.Cc1ccc(CO)cn1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.53
KDM4E B2RXH2 2/20 0.50
L3MBTL1 Q9Y468 2/20 0.50
HDAC1 Q13547 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
CYP4A11 Q02928 2/20 0.46
LOXL2 Q9Y4K0 1/20 0.46
CYP4F2 P78329 1/20 0.45
ALDH1A1 P00352 1/20 0.45
RAB9A P51151 2/20 0.45
GAA P10253 1/20 0.45
TDP1 Q9NUW8 1/20 0.43
MAPT P10636 3/20 0.42
LMNA P02545 1/20 0.42
KMT2A Q03164 1/20 0.42
AR P10275 1/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL64763 0.87 MAPK1 (0.67) MAPK1KDM4EL3MBTL1HDAC1HDAC6
SCHEMBL30574349 0.87 MAPK1 (0.67) MAPK1KDM4EL3MBTL1HDAC1HDAC6
SCHEMBL7362601 0.84 MAPK1 (0.51) MAPK1KDM4EL3MBTL1HDAC1HDAC6
SCHEMBL31029130 0.83 AR (0.52) MAPK1L3MBTL1HDAC1HDAC6CYP4A11
SCHEMBL7528438 0.81 MAPK1 (0.59) MAPK1KDM4EL3MBTL1HDAC1HDAC6
SCHEMBL132853 0.80
SCHEMBL29450844 0.80
SCHEMBL27625609 0.80 MAPK1 (0.57) MAPK1KDM4EL3MBTL1HDAC1HDAC6
Ethyl Acetate SCHEMBL575043 0.79 MAPK1 (0.53) MAPK1KDM4EL3MBTL1HDAC1HDAC6
Hydrochloric Acid SCHEMBL6441917 0.78 TSHR (0.46) KDM4EHDAC1HDAC6ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0631580-A1 PYRIDO 2,3-d]PYRIMIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1995-01-04 EP disclosed
WO-1993019068-A1 PYRIDO[2,3-d]PYRIMIDINE DERIVATIVES AS PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1993-09-30 WO disclosed