SCHEMBL7444366

SCHEMBL7444366

CCc1cc(N(C)c2ccc(-c3ccccc3-c3nnn[nH]3)cc2)n2nc(C(N)=O)cc2n1

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 1/20 0.36
HSD17B10 Q99714 1/20 0.36
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
AHR P35869 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
CHEK2 O96017 1/20 0.32
AGTR1 P30556 1/20 0.30
AGTR2 P50052 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431014 0.93 KDM4E (0.35) KDM4EALDH1A1HSD17B10HPGDMAPT
SCHEMBL7433989 0.87
SCHEMBL7436578 0.86 SMN1; SMN2 (0.31) AGTR1AGTR2
SCHEMBL7440006 0.85 ABCB1 (0.35) KDM4EALDH1A1HPGDMAPTAGTR1
SCHEMBL7448463 0.85 CYP3A4 (0.30)
SCHEMBL7436202 0.85
SCHEMBL7442350 0.85 AGTR1 (0.31) AGTR1AGTR2
SCHEMBL7441331 0.83 HSP90AA1 (0.33) CHEK2
SCHEMBL7433754 0.82 DPP4 (0.41) AGTR1AGTR2
SCHEMBL7444400 0.81 AGTR1 (0.41) KDM4EALDH1A1MAPK1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0628559-B1 Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF LILLY GMBH (DE) 2002-04-03 EP disclosed
US-5602136-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5602137-A Pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1997-02-11 US disclosed
US-5571813-A Fused pyrimidine compounds and their use as pharmaceuticals BEIERSDORF-LILLY GMBH (DE) 1996-11-05 US disclosed
EP-0628559-A1 Pyrimidine compounds and their use as pharmaceuticals Beiersdorf-Lilly GmbH (DE) 1994-12-14 EP disclosed