SCHEMBL7445127

SCHEMBL7445127

O=C(SC(Cc1ccccc1)C(=O)O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MDM2 Q00987 1/20 0.50
CYP1A2 P05177 1/20 0.50
ALPI P09923 1/20 0.47
PKM P14618 1/20 0.47
PTGS1 P23219 1/20 0.47
XIAP P98170 1/20 0.47
SLC7A5 Q01650 1/20 0.47
CPA3 P15088 3/20 0.44
CPA1 P15085 2/20 0.44
FOLH1 Q04609 1/20 0.44
CPB1 P15086 1/20 0.44
CPB2 Q96IY4 1/20 0.44
SRR Q9GZT4 2/20 0.43
SLC1A3 P43003 2/20 0.43
SLC1A2 P43004 2/20 0.43
SLC1A1 P43005 2/20 0.43
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CTRB1 P17538 5/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7164414 1.00 MDM2 (0.50) MDM2CYP1A2ALPIPKMPTGS1
SCHEMBL6990933 1.00 MDM2 (0.50) MDM2CYP1A2ALPIPKMPTGS1
SCHEMBL7449915 0.84 EPHX2 (0.45) CYP1A2CPA1
SCHEMBL7449920 0.84 EPHX2 (0.45) CYP1A2CPA1
SCHEMBL4871578 0.81 POLB (0.51)
SCHEMBL13990223 0.81 POLB (0.51)
SCHEMBL27607672 0.81 POLB (0.51)
SCHEMBL18113160 0.81 MMP8 (0.50) MDM2PKMHSD17B10
SCHEMBL839467 0.80 ALPI (0.53) CYP1A2ALPIPKMPTGS1XIAP
SCHEMBL839468 0.80 ALPI (0.53) CYP1A2ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136842-A INHIBITION OF ENDOTHELIN-CONVERTING ENZYME HOECHST MARION ROUSSEL (FR) 2000-10-24 US disclosed
CN-1218467-A Sulphur derivatives comprising amide bond, method for preparing same, use thereof as drugs, and pharmaceutical compositions containing such derivatives HOEST MARION RUSO S A (FR) 1999-06-02 CN disclosed
WO-1994026719-A1 MERCAPTO-AMIDE DERIVATIVES USEFUL AS NEUTRAL ENDOPEPTIDASE AND ACE INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-11-24 WO disclosed