SCHEMBL7445308

SCHEMBL7445308

CCC(Cc1ccc(C)cc1)c1cc(O)c(C(CC)c2ccc(C)s2)c(=O)o1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.32
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442732 0.94 ESR1 (0.39) CYP2C9ESR1ESR2ALDH1A1MAPT
SCHEMBL7438454 0.93 ESR2 (0.33) CYP2C9ESR1ESR2ALDH1A1MAPT
SCHEMBL7443077 0.93 CYP2C9 (0.37) CYP2C9MAPT
SCHEMBL7443923 0.92 CYP2C9 (0.31) CYP2C9ALDH1A1
SCHEMBL7445588 0.92 MAPT (0.39) CYP2C9ALDH1A1MAPT
SCHEMBL7441942 0.90 MAPT (0.40) ESR1ESR2MAPT
SCHEMBL7446350 0.90
SCHEMBL7441557 0.89 PPARG (0.33)
SCHEMBL7444017 0.87 CYP2C9 (0.31) CYP2C9
SCHEMBL7447190 0.87 CYP2C9 (0.31) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
EP-0668860-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES PHARMACIA & UPJOHN COMPANY (US) 1995-08-30 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed