SCHEMBL7445315

SCHEMBL7445315

CCOC(=O)C(Cc1ccc(-c2ccno2)cc1)N(C)C(=O)c1cc(C)cc(C)c1

nearest known ligand 0.60

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 20/20 0.60
EDNRA P25101 20/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357423 1.00 EDNRB (0.60) EDNRBEDNRA
SCHEMBL7366662 1.00 EDNRB (0.60) EDNRBEDNRA
SCHEMBL7444997 0.89 EDNRB (0.62) EDNRBEDNRA
SCHEMBL7361420 0.89 EDNRB (0.62) EDNRBEDNRA
SCHEMBL7361423 0.89 EDNRB (0.62) EDNRBEDNRA
SCHEMBL7359191 0.83 EDNRB (0.49) EDNRBEDNRA
SCHEMBL7359820 0.80 EDNRB (0.74) EDNRBEDNRA
SCHEMBL7361274 0.79 EDNRB (0.49) EDNRBEDNRA
SCHEMBL7437288 0.79 EDNRB (0.49) EDNRBEDNRA
SCHEMBL7445789 0.77 EDNRB (0.65) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977075-A N-aroylamino acid amides as endothelin inhibitors NOVARTIS AG (CH) 1999-11-02 US disclosed
EP-0821670-A1 N-AROYLAMINO ACID AMIDES AS ENDOTHELIN INHIBITORS Novartis AG (CH) 1998-02-04 EP disclosed
CN-1145075-A Antagonist's of endothelin receptors JAPAT LTD (CH) 1997-03-12 CN disclosed
EP-0753004-A1 ANTAGONISTS OF ENDOTHELIN RECEPTORS Japat Ltd (CH) 1997-01-15 EP disclosed
WO-1996033170-A1 N-AROYLAMINO ACID AMIDES AS ENDOTHELIN INHIBITORS NOVARITS AG (CH) 1996-10-24 WO disclosed
EP-0728145-A1 ENDOTHELIN RECEPTOR ANTAGONISTS Ciba-Geigy Japan Limited (JP) 1996-08-28 EP disclosed
WO-1995026360-A1 ANTAGONISTS OF ENDOTHELIN RECEPTORS JAPAT LTD. (CH) 1995-10-05 WO disclosed
WO-1995012611-A1 ENDOTHELIN RECEPTOR ANTAGONISTS JAPAT LTD. (CH) 1995-05-11 WO disclosed