SCHEMBL7445498

SCHEMBL7445498

COc1cc([C@@H](CC(=O)O)N(C(C)=O)N2C(=O)N[C@](C)(c3ccc(C=NN)cc3)C2=O)cc(OC)c1OC

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
CYP3A4 P08684 2/20 0.33
CYP2C19 P33261 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP2C9 P11712 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
ITGB3 P05106 2/20 0.32
ITGA2B P08514 2/20 0.32
POLB P06746 1/20 0.31
TNF P01375 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPK1 P28482 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446193 0.91 GAA (0.38) CRHBPCRHR2CYP3A4CYP2C19CYP2C9
SCHEMBL7505335 0.90 CYP3A4 (0.35) CRHBPCRHR2CYP3A4CYP2C19KMT2A
SCHEMBL8492985 0.90 CYP3A4 (0.35) CRHBPCRHR2CYP3A4CYP2C19KMT2A
SCHEMBL8490497 0.87 ITGB3 (0.40) CRHBPCRHR2KMT2AMEN1ITGB3
Hydrochloric Acid SCHEMBL8481921 0.86 ITGB3 (0.39) CRHBPCRHR2KMT2AMEN1ITGB3
Acetic Acid SCHEMBL8476499 0.86 ITGB3 (0.39) CRHBPCRHR2KMT2AMEN1ITGB3
Hydrochloric Acid SCHEMBL7438834 0.86 ITGB3 (0.39) CRHBPCRHR2KMT2AMEN1ITGB3
Hydrochloric Acid SCHEMBL7446793 0.86 ITGB3 (0.39) CRHBPCRHR2KMT2AMEN1ITGB3
Hydrochloric Acid SCHEMBL8488366 0.86 ITGB3 (0.39) CRHBPCRHR2KMT2AMEN1ITGB3
SCHEMBL7983484 0.85 ITGB3 (0.46) CYP3A4CYP2C19KMT2ACYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729460-B1 SUBSTITUTED 5-RING HETEROCYCLES, THEIR PREPARATION AND THEIR USE HOECHST AG (DE) 2002-05-15 EP disclosed
WO-1995014008-A1 SUBSTITUTED 5-RING HETEROCYCLES, THEIR PREPARATION AND THEIR USE HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-26 WO disclosed