SCHEMBL7446185

SCHEMBL7446185

COc1ccc(CC(CC2CC2)c2cc(O)c(C(c3cccs3)C3CC3)c(=O)o2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.36
TP53 P04637 2/20 0.35
MAPT P10636 1/20 0.34
MCL1 Q07820 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ALDH1A1 P00352 6/20 0.33
HPGD P15428 2/20 0.32
NQO1 P15559 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
NPC1 O15118 1/20 0.32
POLB P06746 1/20 0.32
RAB9A P51151 1/20 0.32
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439820 0.91 L3MBTL1 (0.37) L3MBTL1TP53MAPTMCL1NPSR1
SCHEMBL7445237 0.91 NQO1 (0.33) ALDH1A1NQO1MAPK1NPC1RAB9A
SCHEMBL7450365 0.90 NQO1 (0.34) NQO1
SCHEMBL7439540 0.90 NQO1 (0.34) NQO1
SCHEMBL7444883 0.89 NQO1 (0.33) TP53NQO1TSHRLMNA
SCHEMBL7450255 0.89 NQO1 (0.33) TP53MAPTNQO1
SCHEMBL7443735 0.88 TP53 (0.35) L3MBTL1TP53MAPTMCL1NPSR1
SCHEMBL7443496 0.87 NQO1 (0.32) NQO1RAB9AHTT
SCHEMBL7442703 0.86 MAPT (0.36) MAPTMCL1POLB
SCHEMBL7443698 0.82 ESR1 (0.35) MAPTALDH1A1HPGDNQO1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0668860-B1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES UPJOHN CO (US) 2002-09-11 EP claimed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO claimed
EP-1203770-A1 Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating hyperplasia and other diseases PHARMACIA & UPJOHN COMPANY (US) 2002-05-08 EP disclosed
WO-1994011361-A1 PYRAN-2-ONES AND 5,6-DIHYDROPYRAN-2-ONES USEFUL FOR TREATING HIV AND OTHER RETROVIRUSES THE UPJOHN COMPANY (US) 1994-05-26 WO disclosed