SCHEMBL7446492

SCHEMBL7446492

Brc1c[c]ccc1CN1CCOCC1

nearest known ligand 0.61

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 7/20 0.61
CYP2C9 P11712 2/20 0.49
ALOX15 P16050 1/20 0.49
HSD17B10 Q99714 1/20 0.49
HRH3 Q9Y5N1 2/20 0.42
HTT P42858 2/20 0.41
ALDH1A1 P00352 3/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
KDM4E B2RXH2 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
CXCR4 P61073 1/20 0.40
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7442877 0.85 TSHR (0.42) CYP2A13ALOX15HRH3HTTALDH1A1
SCHEMBL16462153 0.81 CYP2A13 (0.61) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL16462107 0.81 CYP2A13 (0.61) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL296307 0.79 CYP2A13 (0.63) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL5238359 0.78 HSD17B10 (0.46) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL220727 0.77 HTT (0.48) CYP2A13CYP2C9ALOX15HSD17B10HTT
SCHEMBL16463965 0.77 CYP2A13 (0.45) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL4100083 0.76 CYP2A13 (1.00) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL28805624 0.76 CYP2C9 (0.52) CYP2A13CYP2C9ALOX15HSD17B10HRH3
SCHEMBL6813936 0.75 CYP2A13 (0.96) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed