SCHEMBL16463965

SCHEMBL16463965

FC(F)(F)c1c[c]ccc1CN1CCOCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A13 Q16696 6/20 0.45
CYP2C9 P11712 2/20 0.45
ALOX15 P16050 1/20 0.45
HSD17B10 Q99714 1/20 0.45
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
ATM Q13315 1/20 0.42
HIF1A Q16665 1/20 0.42
EPAS1 Q99814 1/20 0.42
KMT2A Q03164 2/20 0.40
HRH3 Q9Y5N1 1/20 0.39
POLB P06746 1/20 0.39
NR1H2 P55055 1/20 0.39
MEN1 O00255 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27081642 0.86 KDM4E (0.48) ALDH1A1KDM4EATMKMT2APOLB
SCHEMBL1655534 0.82 ALDH1A1 (0.46) CYP2C9ALDH1A1KDM4EATMKMT2A
SCHEMBL28001279 0.82 KDM4E (0.42) ALDH1A1KDM4EATMKMT2AHRH3
SCHEMBL989375 0.82 ALDH1A1 (0.58) ALDH1A1KDM4EATMKMT2APOLB
SCHEMBL16462153 0.80 CYP2A13 (0.61) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL27677146 0.79 ALDH1A1 (0.52) ALDH1A1KDM4EATMKMT2APOLB
SCHEMBL15859936 0.78 KDM4E (0.67) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL16462107 0.77 CYP2A13 (0.61) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL7446492 0.77 CYP2A13 (0.61) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1
SCHEMBL296307 0.75 CYP2A13 (0.63) CYP2A13CYP2C9ALOX15HSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629168-B2 Benzoxazoles and oxazolopyridines being useful as janus kinases inhibitors NOVARTIS AG (CH) 2014-01-14 US claimed
CN-101516860-B Benzoxazoles and oxazolopyridines being useful as FANUS kinases inhibitors NOVARTIS AG 2012-06-27 CN claimed