SCHEMBL7446994

SCHEMBL7446994

O=C1OC(CCc2ccc(F)cc2)(c2ccccc2)CC(O)=C1SCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 5/20 0.44
EGFR P00533 2/20 0.36
CTSB P07858 1/20 0.36
DAO P14920 1/20 0.36
LDHB P07195 1/20 0.35
GAA P10253 2/20 0.35
POLB P06746 1/20 0.35
LMNA P02545 2/20 0.34
ASAH1 Q13510 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAOB P27338 2/20 0.34
PLAAT3 P53816 1/20 0.34
PLAAT5 Q96KN8 1/20 0.34
PLAAT2 Q9NWW9 1/20 0.34
PLAAT4 Q9UL19 1/20 0.34
MAOA P21397 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606612 0.93 LDHA (0.49) LDHAEGFRDAOLDHBGAA
SCHEMBL7446287 0.87 LDHA (0.44) LDHADAOLDHBGAAASAH1
SCHEMBL7446975 0.86 LDHA (0.43) LDHADAOLDHBGAAMAPK1
SCHEMBL6607939 0.85 LDHA (0.50) LDHAEGFRLDHBGAAMAOB
SCHEMBL6603158 0.84 LDHA (0.49) LDHALDHBPLAAT3PLAAT5PLAAT2
SCHEMBL6606818 0.83 LDHA (0.43) LDHADAOPOLBLMNAMEN1
SCHEMBL6605927 0.83 LDHA (0.47) LDHACTSBDAOLDHBLMNA
SCHEMBL6603774 0.83 LDHA (0.48) LDHAEGFRDAOLDHBKMT2A
SCHEMBL7449369 0.83 LDHA (0.44) LDHALDHBLMNAASAH1SMN1; SMN2
SCHEMBL6605273 0.83 HPGD (0.44) LDHAGAALMNAMAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729463-B1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & CO (US) 2002-05-22 EP disclosed
EP-0729464-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1996-09-04 EP disclosed
EP-0729463-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE DAVIS & COMPANY (US) 1996-09-04 EP disclosed
WO-1995014012-A1 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed
WO-1995014011-A2 5,6-DIHYDROPYRONE DERIVATIVES AS PROTEASE INHIBITORS AND ANTIVIRAL AGENTS PARKE, DAVIS & COMPANY (US) 1995-05-26 WO disclosed