SCHEMBL7447216

SCHEMBL7447216

COC(c1ccccc1)C1(C(=O)O)CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
LMNA P02545 3/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
AKR1C1 Q04828 1/20 0.40
CHRM2 P08172 2/20 0.39
CHRM1 P11229 2/20 0.39
CHRM3 P20309 2/20 0.39
CHRM4 P08173 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.37
CYP2C9 P11712 4/20 0.37
CYP3A4 P08684 3/20 0.37
CYP2D6 P10635 3/20 0.37
KDM4E B2RXH2 1/20 0.37
TSHR P16473 2/20 0.36
MAPT P10636 1/20 0.36
CYP2C19 P33261 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
OPRL1 P41146 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16391263 0.92 KMT2A (0.47) KMT2ALMNAMEN1ALDH1A1CYP2C9
SCHEMBL12592080 0.78 AKR1C1 (0.46) KMT2ALMNAMEN1AKR1C1CHRM2
SCHEMBL10233338 0.77 KMT2A (0.43) KMT2ALMNAMEN1ALDH1A1CYP2C9
SCHEMBL12592077 0.75 AKR1C1 (0.47) LMNAAKR1C1CHRM2CHRM1CHRM3
SCHEMBL10408648 0.75 AKR1C1 (0.43) KMT2ALMNAAKR1C1CHRM2CHRM1
SCHEMBL9486483 0.75 AKR1C1 (0.43) KMT2AMEN1AKR1C1CYP2D6NPSR1
SCHEMBL10599613 0.73 CHRM1 (0.40) KMT2ALMNAALDH1A1AKR1C1CHRM1
SCHEMBL12592073 0.72 AKR1C1 (0.42) LMNAAKR1C1CYP2D6NPSR1
SCHEMBL14861334 0.70 CYP2C19 (0.33) KMT2AMEN1KDM4ECYP2C19NPSR1
SCHEMBL517632 0.69 ALOX5 (0.41) KMT2ALMNAALDH1A1AKR1C1CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1005446-A1 N-AROYLPHENYLALANINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-06-07 EP disclosed
WO-1999010313-A1 N-AROYLPHENYLALANINE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1999-03-04 WO disclosed