SCHEMBL7447291

SCHEMBL7447291

N=C(N)NCc1cc(-c2ccc3ccccc3c2)no1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 7/20 0.45
CYP1A2 P05177 4/20 0.45
POLB P06746 2/20 0.44
ALDH1A1 P00352 5/20 0.43
HTT P42858 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
JAK2 O60674 1/20 0.43
LMNA P02545 4/20 0.43
NOTUM Q6P988 2/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 2/20 0.40
TP53 P04637 2/20 0.40
HSD17B10 Q99714 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
SUCNR1 Q9BXA5 3/20 0.39
MAPT P10636 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7447300 0.80 CYP1A2 (0.41) SMN1; SMN2CYP1A2POLBALDH1A1HTT
SCHEMBL189495 0.79 SMN1; SMN2 (0.53) SMN1; SMN2CYP1A2POLBALDH1A1HTT
SCHEMBL7446084 0.78 NOTUM (0.68) SMN1; SMN2CYP1A2ALDH1A1L3MBTL1LMNA
SCHEMBL7440328 0.77 ABCB1 (0.38) SMN1; SMN2CYP1A2ALDH1A1HPGDKDM4E
Hydrochloric Acid SCHEMBL7445767 0.76 ABCB1 (0.38) SMN1; SMN2CYP1A2POLBALDH1A1L3MBTL1
SCHEMBL2840781 0.72 HDAC6 (0.47) SMN1; SMN2CYP1A2POLBALDH1A1HTT
SCHEMBL31686338 0.71 NOTUM (0.58) SMN1; SMN2CYP1A2POLBALDH1A1HTT
SCHEMBL7431655 0.71 S1PR4 (0.38) ALDH1A1KDM4EHSD17B10MEN1KMT2A
SCHEMBL2839518 0.71 HDAC6 (0.47) SMN1; SMN2CYP1A2POLBALDH1A1HTT
SCHEMBL4019637 0.70 IDO1 (0.55) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0397364-B1 HETEROCYCLIC GUANIDINES AS 5HT 3 ANTAGONISTS PFIZER INC. (US) 1993-07-28 EP disclosed
EP-0397364-A1 Heterocyclic guanidines AS 5HT 3 Antagonists PFIZER INC. (US) 1990-11-14 EP disclosed
US-4963689-A ANTIEMETICS, ANALGESICS, GASTROINTESTINAL DISORDERS, SCHIZOPHRENIA PFIZER INC. (US) 1990-10-16 US disclosed