SCHEMBL7440328

SCHEMBL7440328

N=C(N)NCc1ccc(-c2ccc3ccccc3c2)o1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.38
HRH1 P35367 1/20 0.38
F2 P00734 1/20 0.38
PLG P00747 1/20 0.38
PLAU P00749 1/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
PRSS1 P07477 1/20 0.38
CYP1A1 P04798 1/20 0.38
CYP1B1 Q16678 1/20 0.38
NQO2 P16083 1/20 0.38
CYP1A2 P05177 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LDHA P00338 1/20 0.38
LDHB P07195 1/20 0.38
PTPN1 P18031 1/20 0.37
CYP2E1 P05181 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2A6 P11509 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7445767 0.99 ABCB1 (0.38) ABCB1HRH1F2PLGPLAU
SCHEMBL7440332 0.78 HTR6 (0.51) CYP1A2SMN1; SMN2MAPTNPC1TP53
SCHEMBL7447291 0.77 SMN1; SMN2 (0.45) CYP1A2SMN1; SMN2CYP3A4CYP2C9MAPT
Hydrochloric Acid SCHEMBL7445772 0.77 HTR6 (0.50) CYP1A2SMN1; SMN2MAPTNPC1TP53
SCHEMBL7431806 0.76 CYP3A4 (0.65) ABCB1CYP1A1CYP1B1CYP1A2SMN1; SMN2
SCHEMBL7431655 0.74 S1PR4 (0.38) F2PLGPLAUKLKB1KLK1
SCHEMBL30496740 0.72 IDO1 (0.55) F2PLGPLAUKLKB1KLK1
SCHEMBL4019637 0.72 IDO1 (0.55) F2PLGPLAUKLKB1KLK1
SCHEMBL17214863 0.72 ALOX5 (0.50) ABCB1HRH1CYP1A1CYP1B1CYP1A2
SCHEMBL9025706 0.72 LOXL2 (0.54) F2SMN1; SMN2TP53HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0397364-B1 HETEROCYCLIC GUANIDINES AS 5HT 3 ANTAGONISTS PFIZER INC. (US) 1993-07-28 EP disclosed
EP-0397364-A1 Heterocyclic guanidines AS 5HT 3 Antagonists PFIZER INC. (US) 1990-11-14 EP disclosed
US-4963689-A ANTIEMETICS, ANALGESICS, GASTROINTESTINAL DISORDERS, SCHIZOPHRENIA PFIZER INC. (US) 1990-10-16 US disclosed