SCHEMBL7447786

SCHEMBL7447786

COc1ccc(C(=O)c2ccsc2)cc1Br

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.73
CYP1A2 P05177 4/20 0.64
CYP2C19 P33261 4/20 0.64
CYP2D6 P10635 1/20 0.64
HPGD P15428 1/20 0.64
CYP3A4 P08684 2/20 0.51
CYP2C9 P11712 2/20 0.51
TSHR P16473 1/20 0.51
L3MBTL1 Q9Y468 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
MAPT P10636 4/20 0.47
MAPK1 P28482 1/20 0.47
KMT2A Q03164 3/20 0.46
GLA P06280 1/20 0.46
TUBB4A P04350 2/20 0.46
TUBB P07437 2/20 0.46
TUBA3C P0DPH7 2/20 0.46
TUBA1B P68363 2/20 0.46
TUBA4A P68366 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27630437 0.86 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL7444751 0.84 CYP1A2 (0.53) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL6958930 0.81 SLC22A6 (0.73) ALDH1A1CYP1A2CYP2C19HPGDCYP3A4
SCHEMBL28902774 0.80 ALDH1A1 (0.81) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL15947114 0.80 ALDH1A1 (0.86) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL31516304 0.80 ALDH1A1 (0.86) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL25304403 0.78 ALDH1A1 (0.83) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL1818634 0.78 CYP1A2 (1.00) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL15948918 0.78 ALDH1A1 (0.83) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD
SCHEMBL31061882 0.78 ALDH1A1 (0.83) ALDH1A1CYP1A2CYP2C19CYP2D6HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863755-A4 ANTITHROMBOTIC DIAMINES LILLY CO ELI (US) 1999-01-20 EP disclosed
EP-0863755-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1998-09-16 EP disclosed
WO-1997025033-A1 ANTITHROMBOTIC DIAMINES ELI LILLY AND COMPANY (US) 1997-07-17 WO disclosed