Proline

Proline

SCHEMBL7447947

O=C(O)[C@@H]1CCCN1.O=C(O)[C@H]1NCCC1c1ccccc1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC5A2

The experimentally established mechanism targets of Proline. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
BLM P54132 1/20 0.42
KMT2A Q03164 1/20 0.42
ELANE P08246 1/20 0.40
DPP4 P27487 2/20 0.39
ADAM10 O14672 1/20 0.39
ERBB2 P04626 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
RIPK1 Q13546 1/20 0.39
ANPEP P15144 1/20 0.39
CTSC P53634 1/20 0.38
SCN4A P35499 1/20 0.38
SLC1A2 P43004 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16056887 0.88 MEN1 (0.50) MEN1BLMKMT2AADAM10ERBB2
SCHEMBL851578 0.88 MEN1 (0.50) MEN1BLMKMT2AADAM10ERBB2
SCHEMBL4074609 0.88 MEN1 (0.50) MEN1BLMKMT2AADAM10ERBB2
SCHEMBL4780406 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
SCHEMBL199462 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
SCHEMBL5203561 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
SCHEMBL199463 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
SCHEMBL199461 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
SCHEMBL350996 0.88 SLC1A2 (0.47) MEN1BLMKMT2ASLC1A2
Hydrochloric Acid SCHEMBL2297675 0.86 SLC1A2 (0.46) MEN1BLMKMT2ASLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001971-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP disclosed
WO-1999006432-A1 DIPEPTIDE AND RELATED COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO disclosed