SCHEMBL7448685

SCHEMBL7448685

Cn1ccnc1CSc1ccc(C(=N)N)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
IDO1 P14902 1/20 0.38
PTGIR P43119 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
PRSS1 P07477 4/20 0.36
PRSS2 P07478 2/20 0.36
PRSS3 P35030 2/20 0.36
HDAC1 Q13547 1/20 0.36
ALDH1A1 P00352 4/20 0.36
RAB9A P51151 3/20 0.36
NPC1 O15118 3/20 0.36
MAPT P10636 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
POLB P06746 2/20 0.36
TP53 P04637 1/20 0.36
ALOX12 P18054 1/20 0.36
KDM4E B2RXH2 1/20 0.35
HSP90AA1 P07900 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5657607 0.81 KMT2A (0.41) SMN1; SMN2IDO1MEN1KMT2AALDH1A1
SCHEMBL7167511 0.77 PRSS1 (0.42) SMN1; SMN2MEN1KMT2APRSS1PRSS2
SCHEMBL7444492 0.75 KLK1 (0.55) PRSS1PRSS2PRSS3F2TMPRSS6
SCHEMBL15624790 0.68 PRSS1 (0.50) PTGIRPRSS1PRSS2PRSS3ALDH1A1
SCHEMBL952297 0.66
SCHEMBL23565998 0.66 PRSS1 (0.44) SMN1; SMN2IDO1PTGIRMEN1KMT2A
SCHEMBL19486513 0.65 CA12 (0.49) PTGIRPRSS1PRSS2PRSS3F2
Hydrochloric Acid SCHEMBL23541192 0.65 PRSS1 (0.43) SMN1; SMN2IDO1PTGIRMEN1KMT2A
SCHEMBL5653814 0.65 TLR8 (0.39) MEN1KMT2AALDH1A1RAB9ANPC1
SCHEMBL7448690 0.65 KDM4E (0.43) MEN1KMT2APRSS1PRSS2PRSS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed