SCHEMBL7449075

SCHEMBL7449075

N#Cc1cccc(C=C(C(=O)O)c2cccnc2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
MAPT P10636 1/20 0.49
AKR1C1 Q04828 1/20 0.44
VNN1 O95497 2/20 0.44
P4HB P07237 2/20 0.43
GRM5 P41594 4/20 0.43
FBP1 P09467 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP1A1 P04798 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP1B1 Q16678 1/20 0.43
BRAF P15056 1/20 0.42
APP P05067 1/20 0.42
GAA P10253 1/20 0.42
HCAR3 P49019 1/20 0.42
HCAR2 Q8TDS4 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8646712 1.00 ALDH1A1 (0.49) ALDH1A1MAPTAKR1C1VNN1P4HB
SCHEMBL7449069 1.00 ALDH1A1 (0.49) ALDH1A1MAPTAKR1C1VNN1P4HB
SCHEMBL8648599 0.82 ALDH1A1 (0.42) ALDH1A1MAPTVNN1P4HBGRM5
SCHEMBL8646375 0.81 AKR1C1 (0.68) ALDH1A1MAPTAKR1C1MEN1KMT2A
SCHEMBL8646379 0.81 AKR1C1 (0.68) ALDH1A1MAPTAKR1C1MEN1KMT2A
SCHEMBL8649420 0.81 AKR1C3 (0.56) ALDH1A1MAPTAKR1C1MEN1KMT2A
SCHEMBL8649414 0.81 AKR1C3 (0.56) ALDH1A1MAPTAKR1C1MEN1KMT2A
SCHEMBL622907 0.80 AKR1C1 (0.62) ALDH1A1AKR1C1P4HBFBP1MEN1
SCHEMBL622906 0.80 AKR1C1 (0.62) ALDH1A1AKR1C1P4HBFBP1MEN1
SCHEMBL8645516 0.78 TSHR (0.54) ALDH1A1AKR1C1VNN1P4HBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189879-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2002-03-27 EP disclosed
WO-2000071512-A1 INHIBITORS OF FACTOR Xa COR THERAPEUTICS, INC. (US) 2000-11-30 WO disclosed
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed