SCHEMBL7449207

SCHEMBL7449207

CC(O)Cc1ncc(Nc2cncnc2)c(C(=O)O)n1

nearest known ligand 0.52

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 19/20 0.52
FLT4 P35916 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453420 0.91 PDE10A (0.60) PDE10AFLT4
SCHEMBL15048494 0.81 PDE10A (0.55) PDE10A
SCHEMBL7457191 0.79 PDE10A (0.59) PDE10A
SCHEMBL2161270 0.79 PDE10A (0.58) PDE10A
SCHEMBL7448971 0.77 PDE10A (0.49) PDE10A
SCHEMBL7453820 0.75 PDE10A (0.51) PDE10A
SCHEMBL7453331 0.74 PDE10A (0.58) PDE10A
SCHEMBL7449198 0.73 PDE10A (0.59) PDE10A
SCHEMBL7449158 0.73 TSHR (0.34) PDE10A
SCHEMBL7455525 0.72 PDE10A (0.61) PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2580207-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2013-04-17 EP claimed
WO-2011154327-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-12-15 WO claimed
EP-2580207-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2013-04-17 EP disclosed
WO-2011154327-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-12-15 WO disclosed