SCHEMBL7449158

SCHEMBL7449158

CC(O)Cc1ncc(Br)c(C(=O)O)n1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.34
HCAR2 Q8TDS4 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
PDE10A Q9Y233 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1284339 0.80 TDP1 (0.37) TSHRHCAR2TDP1MEN1KMT2A
SCHEMBL6866135 0.78 ALDH1A1 (0.32) HCAR2TDP1MEN1KMT2APKM
SCHEMBL2160060 0.76 HCAR2 (0.35) TSHRHCAR2TDP1MEN1KMT2A
SCHEMBL15894461 0.74 RARB (0.43) TSHRHCAR2TDP1MEN1KMT2A
SCHEMBL2159923 0.73 MEN1 (0.33) TDP1MEN1KMT2APDE10A
SCHEMBL7449207 0.73 PDE10A (0.52) PDE10A
SCHEMBL7457865 0.72 TDP1 (0.31) TDP1MEN1KMT2A
SCHEMBL630361 0.71 KMT2A (0.36) HCAR2TDP1MEN1KMT2A
SCHEMBL21884143 0.67 ALDH1A1 (0.34) TSHRHCAR2TDP1MEN1KMT2A
SCHEMBL15963465 0.67 GRM4 (0.41) HCAR2TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2580207-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2013-04-17 EP disclosed
WO-2011154327-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-12-15 WO disclosed