SCHEMBL7449378

SCHEMBL7449378

CCCCCCOC(=O)NC(=N)c1ccc(NCc2nc3c(C)c(OC(=O)N(CCCO)c4ccccc4)ccc3[nH]2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
MAPT P10636 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
CYP1A2 P05177 2/20 0.32
TSHR P16473 1/20 0.32
MASP2 O00187 1/20 0.32
F2 P00734 1/20 0.32
ADRB2 P07550 1/20 0.32
KLK1 P06870 2/20 0.31
KLK5 Q9Y337 2/20 0.31
MEN1 O00255 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
HDAC1 Q13547 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7452110 0.93 NPC1 (0.36) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7448003 0.92 ALDH1A1 (0.38) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7445819 0.92 NPC1 (0.35) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7449027 0.92 ALDH1A1 (0.36) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7449123 0.86 F2 (0.40) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7447386 0.86 NR1I2 (0.35) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7452514 0.85 F2 (0.42) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7446037 0.85 F2 (0.42) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7445500 0.85 F2 (0.42) ALDH1A1NPC1LMNAMAPTMAPK1
SCHEMBL7442445 0.85 F2 (0.42) ALDH1A1NPC1LMNAMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed