SCHEMBL7449804

SCHEMBL7449804

COc1ccc2cnn3c(-c4c(-c5ccccc5)noc4C)nnc3c2c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.44
MAPT P10636 5/20 0.44
TP53 P04637 3/20 0.44
PTGS1 P23219 1/20 0.42
POLB P06746 1/20 0.41
LMNA P02545 2/20 0.41
BRD4 O60885 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
MEN1 O00255 1/20 0.39
MAPK1 P28482 1/20 0.39
STAT1 P42224 1/20 0.39
KMT2A Q03164 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453636 0.93 PTGS2 (0.45) PTGS2MAPTTP53PTGS1POLB
SCHEMBL7450164 0.88 PTGS2 (0.46) PTGS2MAPTPTGS1LMNAALDH1A1
SCHEMBL7459052 0.86 PTGS2 (0.44) PTGS2MAPTPTGS1LMNAALDH1A1
SCHEMBL7455285 0.86 PTGS1 (0.48) PTGS2MAPTPTGS1POLBLMNA
SCHEMBL7456757 0.85 PTGS2 (0.50) PTGS2MAPTPTGS1LMNABRD4
SCHEMBL7458524 0.83 PTGS1 (0.41) PTGS2MAPTPTGS1POLBTSHR
SCHEMBL7458144 0.83 PTGS2 (0.41) PTGS2MAPTPTGS1LMNASMN1; SMN2
SCHEMBL7450436 0.83 PTGS2 (0.41) PTGS2MAPTPTGS1LMNAALDH1A1
SCHEMBL7451498 0.83 PTGS2 (0.41) PTGS2MAPTPTGS1POLBLMNA
SCHEMBL7450672 0.83 PTGS2 (0.41) PTGS2MAPTPTGS1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002081474-A1 TRIAZOLOPHTHALAZINE / QUINOLINE / ISOQUINOLINE DERIVATIVES WHICH ARE LIGANDS FOR GABA-A RECEPTORS CONTAINING THE ALPHA 5 SUBTYPE MERCK SHARP & DOHME LIMITED (GB) 2002-10-17 WO disclosed