SCHEMBL7450332

SCHEMBL7450332

COc1cc2c(Nc3cc(O[Si](c4ccccc4)(c4ccccc4)C(C)(C)C)c(Cl)cc3F)ncnc2cc1OCc1ccsc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 13/20 0.66
FLT1 P17948 6/20 0.66
EGFR P00533 8/20 0.53
MAPK14 Q16539 2/20 0.51
FLT4 P35916 4/20 0.49
FGFR1 P11362 3/20 0.49
FGFR2 P21802 1/20 0.49
FGFR4 P22455 1/20 0.49
FGFR3 P22607 1/20 0.49
EPHB2 P29323 1/20 0.47
EPHA2 P29317 4/20 0.47
EPHB4 P54760 3/20 0.47
GAK O14976 1/20 0.46
RIPK2 O43353 1/20 0.46
SRC P12931 1/20 0.46
NOD1 Q9Y239 1/20 0.46
ERBB2 P04626 3/20 0.45
AURKA O14965 1/20 0.45
INSR P06213 1/20 0.45
FBP1 P09467 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451653 0.92 EGFR (0.59) KDRFLT1EGFRMAPK14FLT4
SCHEMBL7450324 0.84 KDR (0.63) KDRFLT1EGFRMAPK14FLT4
Hydrochloric Acid SCHEMBL7451047 0.84 KDR (0.75) KDRFLT1EGFRMAPK14FLT4
SCHEMBL7460012 0.83 RET (0.55) KDRFLT1EGFRMAPK14FLT4
SCHEMBL7452247 0.83 MAPK14 (0.58) KDRFLT1EGFRMAPK14FLT4
SCHEMBL7455500 0.83 KDR (0.77) KDRFLT1EGFRMAPK14FLT4
Hydrochloric Acid SCHEMBL7455319 0.81 FLT1 (0.98) KDRFLT1EGFRFLT4FGFR1
SCHEMBL6431182 0.81 EGFR (0.54) KDRFLT1EGFRMAPK14FLT4
SCHEMBL7454326 0.80 FLT1 (1.00) KDRFLT1EGFRFLT4FGFR1
SCHEMBL7459846 0.80 FGFR1 (0.68) KDRFLT1EGFRMAPK14FLT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362336-B1 ADMINISTERING A QUINAZOLINE DERIVATIVE TO A WARM-BLOODED ANIMAL FOR PRODUCING AN ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY REDUCING EFFECT ZENECA LIMITED (GB) 2002-03-26 US disclosed
US-20020032208-A1 Chemical compounds ZENECA LIMITED 2002-03-14 US disclosed
EP-0873319-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-07-25 EP disclosed
US-6258951-B1 ANTICANCER, ANTIARTHRITIC AGENTS ZENECA LIMITED (GB) 2001-07-10 US disclosed
US-6071921-A Chemical compounds ZENECA LIMITED (GB) 2000-06-06 US disclosed
US-5962458-A ANGIOGENESIS INHIBITORS, ANTICANCER AGENTS, ANTIDIABETIC AGENTS, SKIN DISORDERS, AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS, VISION DEFECTS ZENECA LIMITED (GB) 1999-10-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032208-A1 Chemical compounds FLT1, CNKSR1, KDR KDR 3/4885FLT1 1/4885EGFR 48/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.