SCHEMBL7450445

SCHEMBL7450445

CCOC(=O)c1ccc(OCC#Cc2ccc(C[C@H](NC(=O)[C@@H]3CCCN3S(=O)(=O)c3ccc(C)cc3)C(=O)O)cc2)cc1.COCC#Cc1ccc(C[C@H](NC(=O)CN(C)S(=O)(=O)c2ccc(C)cc2)C(=O)O)cc1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 5/20 0.49
ITGB1 P05556 10/20 0.43
ITGA5 P08648 4/20 0.43
ITGB7 P26010 1/20 0.42
ITGAV P06756 3/20 0.41
MAPK1 P28482 2/20 0.40
TSHR P16473 2/20 0.40
ITGA2 P17301 1/20 0.39
KMT2A Q03164 1/20 0.38
ALDH1A1 P00352 2/20 0.38
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HCRTR1 O43613 2/20 0.36
HCRTR2 O43614 2/20 0.36
MMP1 P03956 2/20 0.36
MMP13 P45452 2/20 0.36
ADAM17 P78536 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450450 1.00 ITGA4 (0.49) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7511565 0.92 ITGA4 (0.52) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7506837 0.92 ITGA4 (0.52) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7316222 0.90 ITGA4 (0.59) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7316216 0.90 ITGA4 (0.59) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7325796 0.86 MAPK1 (0.48) ITGA4ITGB1MAPK1KMT2AGAA
SCHEMBL7325803 0.86 MAPK1 (0.48) ITGA4ITGB1MAPK1KMT2AGAA
SCHEMBL7507301 0.86 ITGA4 (0.50) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7326267 0.84 ITGA4 (0.60) ITGA4ITGB1ITGA5ITGB7ITGAV
SCHEMBL7326273 0.84 ITGA4 (0.60) ITGA4ITGB1ITGA5ITGB7ITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001972-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 Elan Pharmaceuticals, Inc. (US) 2000-05-24 EP claimed
WO-1999006431-A1 SUBSTITUTED PHENYLALANINE TYPE COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARMACEUTICALS, INC. (US) 1999-02-11 WO claimed