SCHEMBL7455902

SCHEMBL7455902

Cn1ccnc1SCCO

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.50
RAB9A P51151 6/20 0.48
ALDH1A1 P00352 5/20 0.48
NPC1 O15118 5/20 0.48
POLB P06746 3/20 0.48
KMT2A Q03164 3/20 0.48
HPGD P15428 2/20 0.48
MAPT P10636 2/20 0.48
MEN1 O00255 1/20 0.48
TP53 P04637 1/20 0.48
ALOX12 P18054 1/20 0.48
HSD17B10 Q99714 1/20 0.48
SMN1; SMN2 Q16637 5/20 0.47
ALPL P05186 1/20 0.46
ALPG P10696 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GAA P10253 2/20 0.44
PKM P14618 1/20 0.43
RECQL P46063 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7258742 0.90 KDM4E (0.46) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL7456376 0.89 KDM4E (0.48) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL7357438 0.86 KDM4E (0.46) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL24866430 0.82 KDM4E (0.51) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL15219972 0.82 KDM4E (0.51) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL9044947 0.81 KDM4E (0.50) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL72244 0.81 KDM4E (0.50) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL9046684 0.81 KDM4E (0.50) KDM4ERAB9AALDH1A1NPC1POLB
SCHEMBL422525 0.79 KDM4E (0.49) KDM4ERAB9AALDH1A1NPC1POLB
Hydrochloric Acid SCHEMBL8907355 0.79 KDM4E (0.49) KDM4ERAB9AALDH1A1NPC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6362336-B1 ADMINISTERING A QUINAZOLINE DERIVATIVE TO A WARM-BLOODED ANIMAL FOR PRODUCING AN ANTIANGIOGENIC AND/OR VASCULAR PERMEABILITY REDUCING EFFECT ZENECA LIMITED (GB) 2002-03-26 US disclosed
US-20020032208-A1 Chemical compounds ZENECA LIMITED 2002-03-14 US disclosed
EP-0873319-B1 QUINAZOLINE DERIVATIVES ASTRAZENECA AB (SE) 2001-07-25 EP disclosed
US-6258951-B1 ANTICANCER, ANTIARTHRITIC AGENTS ZENECA LIMITED (GB) 2001-07-10 US disclosed
US-6071921-A Chemical compounds ZENECA LIMITED (GB) 2000-06-06 US disclosed
US-5962458-A ANGIOGENESIS INHIBITORS, ANTICANCER AGENTS, ANTIDIABETIC AGENTS, SKIN DISORDERS, AUTOIMMUNE DISEASES, ANTIINFLAMMATORY AGENTS, VISION DEFECTS ZENECA LIMITED (GB) 1999-10-05 US disclosed
EP-0873319-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1998-10-28 EP disclosed
WO-1997022596-A1 QUINAZOLINE DERIVATIVES ZENECA LIMITED (GB) 1997-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032208-A1 Chemical compounds FLT1, CNKSR1, KDR KDM4E 2469/4885RAB9A 1826/4885ALDH1A1 2174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.