SCHEMBL7459372

SCHEMBL7459372

Cc1nccc(-c2ccccc2)c1O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.45
HDAC4 P56524 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
BACE1 P56817 1/20 0.41
TOP2A P11388 1/20 0.41
ESR2 Q92731 1/20 0.41
RPS6KA3 P51812 2/20 0.41
IKBKB O14920 1/20 0.41
CHUK O15111 1/20 0.41
DAPK3 O43293 1/20 0.41
JAK2 O60674 1/20 0.41
PRKD3 O94806 1/20 0.41
MAP4K4 O95819 1/20 0.41
PAK4 O96013 1/20 0.41
CSF1R P07333 1/20 0.41
RET P07949 1/20 0.41
IGF1R P08069 1/20 0.41
FGFR1 P11362 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27586450 0.83 NUDT1 (0.49) PTK2ALDH1A1HPGDHSD17B10MAPT
SCHEMBL6516685 0.82 CHEK1 (0.46) CHEK1RPS6KA3IKBKBCHUKDAPK3
Bromide SCHEMBL28797051 0.80 CHEK1 (0.45) CHEK1RPS6KA3IKBKBCHUKDAPK3
SCHEMBL10199428 0.79 GRM4 (0.58) CHEK1RPS6KA3IKBKBCHUKDAPK3
SCHEMBL9870675 0.78 RECQL (0.43) CHEK1RPS6KA3IKBKBCHUKDAPK3
SCHEMBL13215846 0.78 MKNK1 (0.39) GRM4NPC1RAB9ACYP2A6ERN1
SCHEMBL13215847 0.77 KDM4E (0.46) NPC1RAB9AALDH1A1HPGDHSD17B10
SCHEMBL9870508 0.77 CHEK1 (0.42) CHEK1ESR2RPS6KA3IKBKBCHUK
SCHEMBL25696391 0.76 CHEK1 (0.45) CHEK1RPS6KA3IKBKBCHUKDAPK3
SCHEMBL5532390 0.76 TACR1 (0.51) CHEK1ALDH1A1SMN1; SMN2TACR1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944626-A4 TROPANE DERIVATIVES AND METHOD FOR THEIR SYNTHESIS UNIV GEORGETOWN (US) 2002-09-04 EP disclosed
EP-0944626-A1 TROPANE DERIVATIVES AND METHOD FOR THEIR SYNTHESIS GEORGETOWN UNIVERSITY (US) 1999-09-29 EP disclosed
WO-1998024788-A1 TROPANE DERIVATIVES AND METHOD FOR THEIR SYNTHESIS GEORGETOWN UNIVERSITY (US) 1998-06-11 WO disclosed