SCHEMBL7459593

SCHEMBL7459593

Cc1ccc(O)c(-c2noc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)c(Cl)c23)c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.34
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
MITF O75030 1/20 0.31
HPGD P15428 1/20 0.30
NT5E P21589 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455649 0.90 NPC1 (0.33) NPC1RAB9AMITF
SCHEMBL7459601 0.86 ESR1 (0.38) HSP90AA1NPC1RAB9AMITF
SCHEMBL7458109 0.85 HSP90AA1 (0.39) HSP90AA1NPC1RAB9AMITFHPGD
SCHEMBL7460214 0.85 PTGDR2 (0.36)
SCHEMBL7462086 0.83 PPARG (0.35) HPGD
SCHEMBL7462783 0.82 PPARG (0.34)
SCHEMBL7467902 0.80 PPARG (0.34)
SCHEMBL7460219 0.78 MCL1 (0.36) HPGD
SCHEMBL7462094 0.77 ALDH2 (0.34) HPGD
SCHEMBL7462790 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed