SCHEMBL7459601

SCHEMBL7459601

Cc1cc(-c2noc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)c(Cl)c23)ccc1O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.38
ESR2 Q92731 2/20 0.38
NPC1 O15118 7/20 0.35
RAB9A P51151 6/20 0.35
MITF O75030 1/20 0.33
CASP3 P42574 1/20 0.31
SENP8 Q96LD8 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
COMT P21964 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459593 0.86 HSP90AA1 (0.34) NPC1RAB9AMITFHSP90AA1
SCHEMBL7458121 0.84 ESR1 (0.46) ESR1ESR2NPC1RAB9AMITF
SCHEMBL7455649 0.80 NPC1 (0.33) NPC1RAB9AMITF
SCHEMBL7460219 0.77 MCL1 (0.36) MEN1KMT2A
SCHEMBL7462094 0.76 ALDH2 (0.34) MEN1KMT2A
SCHEMBL7460214 0.75 PTGDR2 (0.36)
SCHEMBL7462790 0.74
SCHEMBL7462086 0.73 PPARG (0.35)
SCHEMBL7458869 0.73 PTGS2 (0.38) ESR1ESR2NPC1RAB9A
SCHEMBL7467907 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed