SCHEMBL7459716

SCHEMBL7459716

CC(C)n1nnc(C2O[C@@H](n3cnc4c(NCc5ccccc5)nc(NCCc5cn(C)cn5)nc43)[C@H](OC=O)C2O)n1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 10/20 0.44
ADORA3 P0DMS8 6/20 0.44
NT5E P21589 4/20 0.43
ACHE P22303 1/20 0.43
PGK1 P00558 3/20 0.43
PGK2 P07205 3/20 0.43
ADORA2B P29275 5/20 0.42
ADORA1 P30542 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7223843 1.00 ADORA2A (0.44) ADORA2AADORA3NT5EACHEPGK1
SCHEMBL7231338 0.96 PGK1 (0.48) ADORA2AADORA3NT5EPGK1PGK2
SCHEMBL7223844 0.95 NT5E (0.44) ADORA2AADORA3NT5EACHEPGK1
SCHEMBL7224964 0.93 PGK1 (0.45) ADORA2AADORA3NT5EACHEPGK1
Formic Acid SCHEMBL7223839 0.92 PGK1 (0.48) ADORA2AADORA3NT5EPGK1PGK2
SCHEMBL7231332 0.91 PGK1 (0.49) ADORA2AADORA3NT5EPGK1PGK2
SCHEMBL7229729 0.91 ADORA2A (0.48) ADORA2AADORA3PGK1PGK2ADORA2B
SCHEMBL5086139 0.91 PGK1 (0.51) ADORA2AADORA3NT5EPGK1PGK2
SCHEMBL7226421 0.90 ADORA2A (0.41) ADORA2AADORA3PGK1PGK2ADORA2B
SCHEMBL7230061 0.89 ADORA2A (0.46) ADORA2AADORA3ADORA2BADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0948509-B1 2-(PURIN-9-YL)-TETRAHYDROFURAN-3,4-DIOL DERIVATIVES GLAXO GROUP LTD (GB) 2002-10-16 EP disclosed