SCHEMBL7459944

SCHEMBL7459944

CNC(=O)c1n[nH]cc1CN

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
YTHDC1 Q96MU7 1/20 0.41
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
PARP1 P09874 1/20 0.32
PIN1 Q13526 1/20 0.32
BRD4 O60885 1/20 0.32
NTRK1 P04629 2/20 0.32
CREBBP Q92793 1/20 0.32
FLT3 P36888 1/20 0.31
CFTR P13569 1/20 0.31
KDM4E B2RXH2 2/20 0.31
CHEK1 O14757 1/20 0.31
RET P07949 1/20 0.31
PDGFRB P09619 1/20 0.31
PIM1 P11309 1/20 0.31
PDGFRA P16234 1/20 0.31
GSK3B P49841 1/20 0.31
RPS6KA3 P51812 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7451996 0.81 KDM4E (0.42) CREBBPKDM4EHPGDTSHRSMN1; SMN2
SCHEMBL7455406 0.78 LCK (0.30)
SCHEMBL3063009 0.77 YTHDC1 (0.41) YTHDC1PARP1PIN1BRD4NTRK1
SCHEMBL13651216 0.75 KDM4E (0.48) KDM4ETSHR
SCHEMBL25086311 0.74 YTHDC1 (0.42) YTHDC1PIN1BRD4CREBBPFLT3
SCHEMBL15186359 0.74 YTHDC1 (0.42) YTHDC1PARP1PIN1BRD4CREBBP
SCHEMBL13816862 0.73 YTHDC1 (0.41) YTHDC1PIN1BRD4CREBBPFLT3
SCHEMBL2385166 0.73 CREBBP (0.42) YTHDC1PIN1BRD4CREBBPCFTR
SCHEMBL15112120 0.70 YTHDC1 (0.39) YTHDC1PIN1CREBBPCHEK1RET
SCHEMBL13543760 0.69 SLC6A2 (0.40) YTHDC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2580207-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. Hoffmann-La Roche AG (CH) 2013-04-17 EP disclosed
WO-2011154327-A1 NITROGEN CONTAINING HETEROARYL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2011-12-15 WO disclosed