SCHEMBL7459997

SCHEMBL7459997

COc1cccc(COc2[c]ccc(-c3ccccc3)c2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.52
HTR1A P08908 3/20 0.47
ABCB1 P08183 2/20 0.47
DRD2 P14416 2/20 0.47
IDO1 P14902 2/20 0.47
AGXT P21549 2/20 0.47
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
BCHE P06276 1/20 0.44
GABRA1 P14867 1/20 0.44
GABRG2 P18507 1/20 0.44
GABRB3 P28472 1/20 0.44
GABRA5 P31644 1/20 0.44
GABRA3 P34903 1/20 0.44
GABRA2 P47869 1/20 0.44
MRGPRX4 Q96LA9 2/20 0.44
NR4A2 P43354 1/20 0.44
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468357 0.84 AGXT (0.43) MAOBIDO1AGXTGABRG2GABRB3
SCHEMBL6810250 0.82 MAOB (0.55) MAOBHTR1AABCB1DRD2IDO1
SCHEMBL2202368 0.82 MAOB (0.58) MAOBHTR1AABCB1DRD2BCHE
SCHEMBL7464303 0.81 MAOB (0.44) MAOBIDO1AGXTMRGPRX4NR4A2
SCHEMBL13722545 0.81 MAOB (0.61) MAOBHTR1AABCB1DRD2IDO1
SCHEMBL7464222 0.78 FFAR1 (0.41) MAOBIDO1AGXTHTTSMN1; SMN2
SCHEMBL27589325 0.77 CYP3A4 (0.50) MAOBABCB1
SCHEMBL13263642 0.76 MAOB (0.79) MAOBHTR1AABCB1DRD2IDO1
SCHEMBL7460676 0.76 KDM4E (0.49) HTR1AABCB1IDO1ADRA1DADRA1A
SCHEMBL7461083 0.75 MAOB (0.51) MAOBHTR1AABCB1DRD2IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed