SCHEMBL7463226

SCHEMBL7463226

COc1ccccc1C(Oc1c[c]ccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.51
TDO2 P48775 1/20 0.51
CYP19A1 P11511 1/20 0.35
MEN1 O00255 6/20 0.35
KMT2A Q03164 6/20 0.35
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
MAPK1 P28482 1/20 0.35
HTT P42858 1/20 0.35
PBRM1 Q86U86 1/20 0.35
SLC6A2 P23975 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7466396 0.89 CYP2D6 (0.43) IDO1TDO2MEN1KMT2AMAPK1
SCHEMBL7466298 0.85 IDO1 (0.37) IDO1TDO2MEN1KMT2AMAPK1
SCHEMBL7461466 0.84 PBRM1 (0.47) ALDH1A1L3MBTL1PBRM1SRD5A2CA4
SCHEMBL7466782 0.83 SRD5A2 (0.45) IDO1TDO2PBRM1TSHRSLC6A4
SCHEMBL7461173 0.81 IDO1 (0.50) IDO1TDO2MEN1KMT2AALDH1A1
SCHEMBL7461086 0.80 CASR (0.42) L3MBTL1PBRM1SRD5A2
SCHEMBL7470957 0.78 IDO1 (0.43) IDO1TDO2OPRM1OPRD1SLC6A2
SCHEMBL7455793 0.78 SRD5A2 (0.39) IDO1TDO2KMT2AALDH1A1HTT
SCHEMBL7460080 0.75 IDO1 (0.49) IDO1TDO2MEN1KMT2AOPRM1
SCHEMBL7456441 0.74 IDO1 (0.54) IDO1TDO2CYP19A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP claimed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO claimed