SCHEMBL7463303

SCHEMBL7463303

NC(=O)C(Br)c1cccc(F)c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC5 Q9UQL6 1/20 0.50
CES2 O00748 2/20 0.49
CES1 P23141 2/20 0.49
PARP1 P09874 1/20 0.48
KCNN4 O15554 3/20 0.44
IDO1 P14902 1/20 0.42
TDO2 P48775 1/20 0.42
CNR2 P34972 1/20 0.42
PKM P14618 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4390797 0.85 HDAC4 (0.53) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL29530737 0.85 HDAC4 (0.53) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL9298252 0.85 HDAC4 (0.53) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL307849 0.82 HDAC4 (0.55) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL29531136 0.81 HDAC4 (0.50) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL9298392 0.81 HDAC4 (0.50) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL9298388 0.81 HDAC4 (0.50) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL7680152 0.80 CES2 (0.44) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL1354521 0.79 HDAC4 (0.51) EPHX1HDAC4HDAC7HDAC5CES2
SCHEMBL1354525 0.79 HDAC4 (0.51) EPHX1HDAC4HDAC7HDAC5CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077701-A4 ANTI-VIRAL COMPOUNDS LILLY CO ELI (US) 2002-03-20 EP disclosed
US-6358971-B1 FOR INHIBITING THE GROWTH OF A PICORNAVIRUS ELI LILLY AND COMPANY 2002-03-19 US disclosed
CN-1292697-A Anti-viral compound LILLY CO ELI (US) 2001-04-25 CN disclosed
EP-1077701-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 2001-02-28 EP disclosed
WO-1999059587-A1 ANTI-VIRAL COMPOUNDS ELI LILLY AND COMPANY (US) 1999-11-25 WO disclosed