SCHEMBL746352

SCHEMBL746352

COCCNS(=O)(=O)N1CCC2(CCN(c3ccc(OC(F)(F)F)cc3)C2=O)CC1

nearest known ligand 0.58

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 19/20 0.58
METAP2 P50579 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3744928 0.90 LIPE (0.65) LIPE
SCHEMBL744442 0.88 LIPE (0.62) LIPE
SCHEMBL747135 0.83 LIPE (0.64) LIPE
SCHEMBL746965 0.82 LIPE (0.62) LIPE
SCHEMBL744562 0.81 LIPE (0.69) LIPE
SCHEMBL745817 0.81 LIPE (0.58) LIPE
SCHEMBL744233 0.80 LIPE (0.55) LIPE
SCHEMBL746001 0.80 LIPE (0.74) LIPEMETAP2
SCHEMBL1589353 0.80 LIPE (0.80) LIPE
SCHEMBL1589383 0.80 LIPE (0.64) LIPEMETAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8329904-B2 Azacyclic derivatives HOFFMANN-LA ROCHE INC. (US) 2012-12-11 US disclosed
US-8329904-B2 Azacyclic derivatives HOFFMANN-LA ROCHE INC. (US) 2012-12-11 US disclosed
EP-2430023-A1 AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-21 EP disclosed
WO-2010130665-A1 AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2010-11-18 WO disclosed